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醫藥化工出口貿易
Pharmaceutical export trade

Intermediates 

醫藥中間體
NO. Product name Classification CAS NO.
1 Methyl 4-amino-5-ethylsulfonyl-2-methoxybenzoate Amisulpride 80036-89-1
2 4-Amino-5-ethylsulfonyl-2-methoxybenzoic acid Amisulpride 71675-87-1
3 2-Chloro-1,4-naphthoquinone Atovaquone 1010-60-2
4 4-(4-Chlorophenyl)cyclohexanecarboxylic acid Atovaquone 49708-81-8
5 4-Chloro-7-((2-(trimethylsilyl)ethoxy)methyl-7H-pyrrolo[2,3-d]pyrimidine Bricitinib 941685-26-3
6 1-(1-ethoxyethyl)-4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H pyrazole Bricitinib 1029716-44-6
7 2-(1-(ethylsulfonyl)azetidin-3-ylidene)acetonitrile Bricitinib 1187595-85-2
8 N-(5-chloropyridin-2-yl)-5-methoxy-2-nitrobenzamide Betrixaban 280773-16-2
9 2-Amino-N-(5-chloropyridin-2-yl)-5-methoxybenzamide Betrixaban 280773-17-3
10 4-Cyanobenzoic acid. Betrixaban 619-65-8
11 5-methoxy-2-nitrobenzoic acid Betrixaban 1882-69-5
12 4-Nitrobenzyl(2S,4S)-4-acetylthio-2-[[N-sulfamoyl-N-(tertbutoxycarbonyl)amino]methyl]pyrrolidine-1-carboxylate(Doripenem side-chain) Doripenem 491878-06-9
13 (R)-3-AMINO-1-BUTANOL Dolutegravir 61477-40-5
14 2,4-Difluorobenzylamine Dolutegravir 72235-52-0
15 (3S)-3-[4-[(2-Chloro-5-iodophenyl)methyl]phenoxy]tetrahydro-furan Empagliflozin 915095-94-2
16 (3S)-3-[4-[(5-Bromo-2-chlorophenyl)methyl]phenoxy]tetrahydro-furan Empagliflozin 915095-89-5
17 2-Amino-4,5-bis(2-methoxyethoxy)benzoic acid ethyl ester hydrochloride Erlotinib 183322-17-0
18 6,7-bis-(2-Methoxyethoxy)-quinazolin-4(3h)-one Erlotinib 179688-29-0
19 4-chloro-6,7-bis(2-methoxyethoxy)-4(3H)-quinazoline Erlotinib 183322-18-1
20 3-Ethynylbenzenamine hydrochloride Erlotinib 207226-02-6
21 (5R,6S,8R,2R)-2-(2-Tetrahydrofuryl)6-hydroxyethylpenem-3-carboxylate monosodium salt Faropenem 58365-51-6/ 120705-67-1
22 2'-Deoxy-2,2'-difluoro-D-erythro-pentofuranous-1-ulose-3,5-dibenzoate Gemcitabine 122111-01-7
23 2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate-1-methanesulfonate Gemcitabine 134877-42-2
24 2’,2’-Difluoro-2'-deoxycyodine-3',5'-dibenzoate Gemcitabine 134790-39-9
25 Gemcitabine base Gemcitabine 95058-81-4
26 4-chloro-7-methoxyquinoline-6-carboxamide Lenvatinib 417721-36-9
27 1,4-dihydro-7-methoxy-4-oxo-6-quinolinecarboxylic acid methyl ester Lenvatinib 205448-65-3
28 Methyl 4-chloro-7-methoxyquinoline-6-carboxylate Lenvatinib 205448-66-4
29 [2-(Methylamino)-3-pyridyl]methanol Isavuconazole 32399-12-5
30 (as,βr)-β-(2,5-difluorophenyl)-β-hydroxy-a-methyl-1h-1,2,4-triazole-1- butanenitrile Isavuconazole 241479-74-3
31 Shikimic acid Oseltamivir 138-59-0
32 (1S,5R,6S)-Ethyl-5-(pentan-3-yl-oxy)-7-oxa-bicyclo[4.1.0]hept-3-ene-3- carboxylate Oseltamivir 204254-96-6
33 2-Chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one Palbociclib 1013916-37-4
34 href="http://www.shentong88.cn/pro_detail/id/197"6-Bromo-2- chloro-8-cyclopentyl-5-methylpyrido[2,3-d]pyrimidin-7(8H)-one Palbociclib 1016636-76-2
35 4-(6-Aminopyridin-3-yl)piperazine-1-carboxylic acid tert-butyl ester Palbociclib 571188-59-5
36 (5R-cis)-Toluene-4-sulfonic acid 5-(2,4-difluorophenyl)-5-(1H-1,2,4- triazol-1-yl)methyltetrahydrofuran-3-ylmethyl ester (Chain A) Posaconazole 149809-43-8
37 2-[(1S,2S)-1-Ethyl-2-bezyloxypropyl]-2,4-dihydro-4-[4-[4-(4-hydroxyphenyl)-1-piperazinyl]phenyl]-3H-1,2,4-triazol-3-one (ChainB+Chain C) Posaconazole 184177-83-1
38 (2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)aMino)-2- Methylpentanoic acid Sacubitril 1012341-50-2
39 (2R,4S)-Ethyl 5-([1,1'-biphenyl]-4-yl)-4-amino-2-methylpentanoate nydrochloride Sacubitril 149690-12-0
40 (1S,3S,5S)-3-(AMinocarbonyl)-2-azabicyclo[3.1.0]hexane-2-carboxylic acid tert-butyl ester Saxagliptir 361440-67-7
41 Boc-3-Hydroxy-1-adamantyl-D-glycine Saxagliptir 361442-00-4
42 N-(2-(Diethylamino)ethyl)-5-formyl-2,4-dimethyl-1H-pyrrole-3- carboxamide Sunitinib 356068-86-5
43 5-Formyl-2,4-dimethyl-1H-pyrrole-3-carboxylic acic Sunitinib 253870-02-9
44 Ethyl 5-formyl-2,4-dimethyl-1H-pyrrole-3-carboxylate Sunitinib 2199-59-9
45 5-Fluoro-2-oxindole Sunitinib 56341-41-4
46 (2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a] pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)but-2-en-2-amine Sitagliptin 767340-03-4
47 (2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a] pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-one Sitagliptin 764667-65-4
48 3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride Sitagliptin 762240-92-6
49 Boc-(R)-3-Amino-4-(2,4,5-trifluorophenyl)butanoic acid Sitagliptin 486460-00-8
50 2,4,5-Trifluorophenylacetic acid Sitagliptin 209995-38-0
51 5-Amino-4-imidazolecarboxamide Temozolomide 360-97-4
52 4-Amino-5-imidazolecarboxamide hydrochloride Temozolomide 72-40-2
53 4-Chloropyrrolo[2,3-d]pyrimidine Tofacitinib 3680-69-1
54 (3R,4R)-1-Benzyl-N,4-dimethylpiperidin-3-amine dihydrochloride Tofacitinib 1062580-52-2
55 4-Chloro-6-ethyl-5-fluoropyrimidine Voriconazole 137234-74-3
56 (2R,3S/2S,3R)-3-(4-Chloro-5-fluoro-6-pyrimidinyl)-2-(2,4-difluorophenyl)- 1-(1H-1,2,4-triazol-1-yl)-2-butanol hydrochloride(N-2 step Voriconazole 188416-35-5
57 (2R,3S/2S,3R)-2-(2,4-difluorophenyl)-3-(5-fluoro-4-pyrimidinyl)-1-(1H- 1,2,4-triazol-1-yl)-2-butanol (N-1step) Voriconazole 182230-43-9
58 Tetrabenzyl-voglibose Voglibose 115250-39-0
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